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Aqueous Fraction from Hibiscus sabdariffa Relaxes Mesenteric Arteries of Normotensive and Hypertensive Rats through Calcium Current Reduction and Possibly Potassium Channels Modulation

Anas M A Alsayed , Bei Li Zhang , Pierre Bredeloux , Leslie Boudesocque-Delaye , Angèle Yu , et al.
Nutrients, 2020, 12 (6), pp.E-1782. ⟨10.3390/nu12061782⟩
Journal articles hal-02881241v1
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Synthesis of Alkyl-Glycerolipids Standards for Gas Chromatography Analysis: Application for Chimera and Shark Liver Oils

Michelle Pinault , Cyrille Guimaraes , Hélène Couthon , Jérôme Thibonnet , Delphine Fontaine , et al.
Marine drugs, 2018, 16 (4), ⟨10.3390/md16040101⟩
Journal articles hal-01744078v1

Monitoring the water content in NADES extracts from spirulina biomass by means of ATR-IR spectroscopy

Suha Elderderi , Soukaina Hilali , Laura Wils , Igor Chourpa , Martin Soucé , et al.
Analytical Methods, 2022, ⟨10.1039/D2AY00234E⟩
Journal articles hal-03662550v1
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Preparation of 3‐Alkylidenephthalides: Recent Advances

Julien Petrignet , Jérôme Thibonnet , Laurent Commeiras , David Gueyrard
European Journal of Organic Chemistry, 2022, 2022 (22), ⟨10.1002/ejoc.202200344⟩
Journal articles hal-03862612v1
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Synthesis and biological evaluation of 3,4-dihydro-1H-[1,4] oxazepino [6,5,4-hi] indol-1-ones and 4,6-dihydrooxepino [5,4,3-cd] indol-1(3H)-ones as Mycobacterium tuberculosis inhibitors

Bastien Champciaux , Clément Raynaud , Albertus Viljoen , Loïc Chene , Jérôme Thibonnet , et al.
Bioorganic & Medicinal Chemistry Letters, 2021, 43, pp.116248. ⟨10.1016/j.bmc.2021.116248⟩
Journal articles hal-03588623v1

In Situ Water Quantification in Natural Deep Eutectic Solvents Using Portable Raman Spectroscopy

Suha Elderderi , Laura Wils , Charlotte Leman-Loubière , Hugh Byrne , Igor Chourpa , et al.
Molecules, 2021, 26 (18), pp.5488. ⟨10.3390/molecules26185488⟩
Journal articles hal-03346166v1
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Efficient One-Pot Synthesis of Triazole-Linked Morpholinone Scaffolds by CuAAC in the Presence of 18-Crown-6

A. Mayooufi , M. Romdhani-Younes , Jérôme Thibonnet
SynOpen, 2018, 02 (04), pp.0298-0305. ⟨10.1055/s-0037-1610399⟩
Journal articles hal-02172433v1
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Straightforward Access to a Great Diversity of Complex Biorelevant γ-Lactams Thanks to a Tunable Cascade Multicomponent Process

Muhammad Idham Darussalam Mardjan , Atef Mayooufi , Jean-Luc Parrain , Jérôme Thibonnet , Laurent Commeiras
Illustration. France. 2020
Image hal-02873547v1
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Lupin (Lupinus spp.) seeds exert anthelmintic activity associated with their alkaloid content

O. Dubois , C. Allanic , C. L Charvet , F. Guégnard , H. Février , et al.
Scientific Reports, 2019, 9 (1), 12 p. ⟨10.1038/s41598-019-45654-6⟩
Journal articles hal-02176665v1
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Natural Deep Eutectic Solvents as sustainable solvent for Suzuki-Miyaura cross- coupling reactions applied to imidazo-fused heterocycles

Pierre-Olivier Delaye , Mélanie Pénichon , Leslie Boudesocque-Delaye , Cécile Enguehard-Gueiffier , Alain Gueiffier
SynOpen, 2018, 2 (04), pp.306 - 311. ⟨10.1055/s-0037-1610400⟩
Journal articles hal-02172280v1
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Bioinspired imidazo[1,2-a:4,5-c’]dipyridines with dual antiproliferative and anti-migrative properties in human cancer cells: The SAR investigation

Abdulrahim Alzain , Lucie Brisson , Pierre-Olivier Delaye , Mélanie Pénichon , Stéphanie Chadet , et al.
European Journal of Medicinal Chemistry, 2021, 218, pp.113258. ⟨10.1016/j.ejmech.2021.113258⟩
Journal articles hal-03202963v1
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Synthèse de la Cytosporone E et analogues

Emilie Thiery , Walaa Baderaldeen , Virginie Herve , Emilie Camiade , Jérôme Thibonnet , et al.
8ème Symposium Francophone de Synthèse Totale (SFST8), May 2018, Bordeaux, France. 2018
Conference poster hal-01822886v1
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Preparation of 3‐Alkylidenephthalides: Recent Advances

Julien Petrignet , Jérôme Thibonnet , Laurent Commeiras , David Gueyrard
France. 2022
Image hal-03862716v1
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Total synthesis of enhygrolide A and analogs

Douha Sghairi , Moufida Romdhani-Younes , Vincent Guilloteau , Julien Petrignet , Jérôme Thibonnet
Tetrahedron Letters, 2020, 61, pp.151786 -. ⟨10.1016/j.tetlet.2020.151786⟩
Journal articles hal-03489593v1
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Spirulina platensis sustainable lipid extracts in alginate-based nanocarriers: An algal approach against biofilms

R. Boutin , E. Munnier , N. Renaudeau , M. Girardot , M. Pinault , et al.
Algal Research - Biomass, Biofuels and Bioproducts, 2019, 37, pp.160-168. ⟨10.1016/j.algal.2018.11.015⟩
Journal articles hal-01955429v1

Improved Condensation of 2-pyridyllithium Intermediates with Aldehydes: Application for the Synthesis of 2-(polyhydroxyalkyl)pyridines

Corinne Comoy , Julien Petrignet , Estelle Banaszak , Anthony Chartoire , Yves Fort
Letters in Organic Chemistry, 2009, 6 (1), pp.50-56. ⟨10.2174/157017809787003214⟩
Journal articles hal-02186916v1
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Gold-silver catalyzed straightforward one pot synthesis of pyrano[3,4- b]pyrrol-7(1H)-ones

P.-O Delaye , J. Petrignet , Emilie Thiery , J Thibonnet
Organic & Biomolecular Chemistry, 2017, 15 (35), pp.7290-7295. ⟨10.1039/c7ob01849e⟩
Journal articles hal-02170750v1

Development of a bio­active fluorescent inhibitor probe targeting the Rho kinase ROCK for monitoring inhibition action

Justine Corret , Sokaina Hammoud , Frédéric Buron , Pierre Daligaux , Christophe Chesné , et al.
FEBS 2021, the 45th FEBS Congress, Jul 2021, Lnubljana, virtual, Slovenia
Conference poster hal-03679980v1
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Synthesis and Reactivity of Oxazinoindolones via Regioselective 6- exo-dig Iodolactonization Reaction

Sokaina Hammoud , Elsa Anselmi , Khalil Cherry , Jean-Claude Kizirian , Jérôme Thibonnet
European Journal of Organic Chemistry, 2018, 2018 (45), pp.6314-6327. ⟨10.1002/ejoc.201801167⟩
Journal articles hal-02172429v1
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Emergence of Copper-mediated formation of C-C bonds

Carine Maaliki , Emilie Thiery , Jérôme Thibonnet
European Journal of Organic Chemistry, 2017, 2017 (2), pp.209-228. ⟨10.1002/ejoc.201600540⟩
Journal articles hal-01601331v1
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Glycerol-based NaDES as green solvents for ultrasound-assisted extraction of phycocyanin from Arthrospira platensis—RSM optimization and ANN modelling

Soukaina Hilali , Laura Wils , Alia Chevalley , Barbara Clement-Larosière , Leslie Boudesocque-Delaye
Biomass Conversion and Biorefinery, 2022, ⟨10.1007/s13399-021-02263-6⟩
Journal articles hal-03547594v1
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Synthesis and evaluation of heterocycle structures as potential inhibitors of Mycobacterium tuberculosis UGM

Carine Maaliki , Jian Fu , Sydney Villaume , Albertus Viljoen , Clément Raynaud , et al.
Bioorganic and Medicinal Chemistry, 2020, 28 (13), pp.115579. ⟨10.1016/j.bmc.2020.115579⟩
Journal articles inserm-03082669v1
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Crystalline tetrazepam as a case study on the volume change on melting of molecular organic compounds

Ivo Rietveld , Philippe Négrier , Maria Barrio , Hassan Allouchi , René Ceolin , et al.
International Journal of Pharmaceutics, 2020, 593, pp.120124. ⟨10.1016/j.ijpharm.2020.120124⟩
Journal articles hal-03053325v1

Synthesis, antibacterial and cytotoxic evaluation of cytosporone E and analogs

Walaa Ibraheem , Capucine Chaar , Emilie Camiade , Virginie Hervé , Delphine Fouquenet , et al.
Journal of Molecular Structure, 2022, 1252, 12 p. ⟨10.1016/j.molstruc.2021.132135⟩
Journal articles hal-03509478v1

On the Dimorphism and the Pressure-Temperature State Diagram of Gestodene, a Steroidal Progestogen Contraceptive

Ivo B. Rietveld , Hassan Allouchi , René Ceolin
57th EHPRG Meeting on High pressure science and technology, Sep 2019, Prague, Czech Republic
Conference poster hal-02352383v1

Development of new highly potent imidazo[1,2-b]pyridazines targeting Toxoplasma gondii calcium-dependent protein kinase 1

Espérance Moine , Isabelle Dimier-Poisson , Cécile Enguehard-Gueiffier , Cédric Logé , Mélanie Pénichon , et al.
European Journal of Medicinal Chemistry, 2015, 105, pp.80-105. ⟨10.1016/j.ejmech.2015.10.004⟩
Journal articles hal-02389861v1
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A network of weak hydrogen bonds in the crystal structure of Tetrazepam

H. Allouchi , R. Ceolin , A. Gueiffier , Ivo B. Rietveld
Annales Pharmaceutiques Françaises, 2019, 77 (2), pp.121-125. ⟨10.1016/j.pharma.2018.11.002⟩
Journal articles hal-02147887v1
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Easy installation of 1,2,3-triazoles or iodo-1,2,3-triazoles onto indole-fused oxazinones via CuAAC-based MCR in the presence of 18-crown-6

A Mayooufi , M Romdhani-Younes , Y Carcenac , Jérôme Thibonnet
Synthetic Communications, In press, ⟨10.1080/00397911.2019.1611857⟩
Journal articles hal-02172442v1

Development of a bio­active fluorescent inhibitor probe targeting the Rho kinase ROCK for monitoring inhibition action

Justine Corret , Sokaina Hammoud , Frédéric Buron , Pierre Daligaux , Christophe Chesné , et al.
FEBS 2021, the 45th FEBS Congress, Jul 2021, Virtual, France
Conference papers hal-03668584v1

Cassia sieberiana root bark used in traditional medicine in Togo: Anthelmintic property against Haemonchus contortus and tannins composition

Iwaba Kpabi , Thibaut Munsch , Amégninou Agban , Isabelle Théry-Koné , Joelle Dorat , et al.
South African Journal of Botany, 2022, 151 (part B), pp.549-558. ⟨10.1016/j.sajb.2022.05.055⟩
Journal articles hal-03918718v1